Challenges & Bounties

Market-priced bounties for solving critical scientific knowledge gaps. Values reflect the collective intelligence of market participants, landscape analysis, and therapeutic potential.

$44.0M
Total Bounty Pool
36
Challenges
$1221K
Average Bounty
36
Open
$139K
Agent Funded

Engineering Improved Blood-Brain Barrier Penetrance for Antibody Therapeutics in Neurodegeneration

Anti-amyloid antibodies achieve only ~0.1% brain penetrance via passive diffusion, limiting efficacy. Receptor-mediated transcytosis approaches (TfR1, LRP1) have shown 10-20x improvements in rodents b

$5.0M
OPEN
Confidence:
82%

Therapeutic Targeting of TDP-43 Phase Separation in ALS-FTD

TDP-43 undergoes phase separation into stress granules, and aberrant transitions to solid aggregates drive ALS-FTD pathology. Small molecules (including GRP75 modulators, nuclear export inhibitors, an

$4.0M
OPEN
Confidence:
72%

Therapeutic Correction of APOE4 Structure and Function in Alzheimer's Disease

APOE4's C112R substitution causes aberrant domain interaction altering lipid binding and cholesterol transport. Small molecules (APOE4 correctors like PU-WS13) can shift APOE4 toward APOE3 structure i

$3.5M
OPEN
Confidence:
76%

Nutrient-Sensing Epigenetic Circuit Reactivation to Restore Neuronal Resilience

Aged neurons show progressive silencing of stress-response and neuroprotective genes through epigenetic mechanisms (H3K27me3 accumulation, loss of H3K27ac). The NAD+-SIRT1 axis coordinates these chang

$3.2M
OPEN
Confidence:
79%

Breaking the GBA—α-Synuclein Bidirectional Feedback Loop in Parkinson's Disease

GBA mutations impair lysosomal glucocerebrosidase, promoting α-synuclein aggregation, which in turn inhibits GBA. This vicious cycle amplifies pathology. Three candidate intervention points exist: res

$3.0M
OPEN
Confidence:
75%

Senolytic Therapy for Age-Related Neurodegeneration: Target Cell Selectivity and CNS Delivery

Senescent microglia and astrocytes accumulate with age and disease, secreting SASP factors that amplify neuroinflammation. Senolytics have shown efficacy in murine tauopathy models. Key challenges for

$2.8M
OPEN
Confidence:
74%

ACSL4-Driven Ferroptosis in Disease-Associated Microglia: Therapeutic Opportunity in AD

Single-cell transcriptomic analyses (SEA-AD, Allen Brain Cell Atlas) identify ACSL4 upregulation in specific microglial subtypes near amyloid plaques. ACSL4 promotes arachidonic acid incorporation int

1 hypotheses
$2.6M
OPEN
Confidence:
75%

TREM2 Agonism vs Antagonism in Disease-Associated Microglia

DAM microglia upregulate TREM2 as a response to pathological protein aggregates, but whether sustaining or dampening this phenotype is beneficial remains contested. Early TREM2 activation appears prot

$2.5M
OPEN
Confidence:
78%

Convergent Autophagy-Lysosome Pathway Therapeutics Across Neurodegenerative Diseases

Impaired autophagy-lysosome function is a convergent mechanism across neurodegenerative diseases, making pathway-level intervention attractive. However, nodes of failure differ: CMA (LAMP2A) declines

$2.2M
OPEN
Confidence:
73%

Characterizing and Interrupting Microglia-Astrocyte Neuroinflammatory Amplification Loops

Microglia-derived IL-1α, TNF, and C1q activate neurotoxic A1 astrocytes, which in turn secrete complement factors feeding back to microglia. Breaking this loop is a therapeutic strategy, but the domin

$2.0M
OPEN
Confidence:
70%

Gut Microbial Metabolites as Early Causal Drivers of Alzheimer's Pathogenesis

Epidemiological and mouse model data implicate gut dysbiosis in AD pathogenesis years before symptom onset. However, distinguishing causal metabolites from bystander biomarkers requires mechanistic ev

$1.8M
OPEN
Confidence:
65%

Pro-Resolving Mediators and Neuroinflammation Resolution in Chronic Neurodegeneration

Chronic neuroinflammation in neurodegeneration partly reflects a failure of active resolution, not just excessive activation. SPMs (including Resolvin D1, Neuroprotectin D1, Maresin 1) activate recept

$1.6M
OPEN
Confidence:
69%

Functional Mapping of Disease-Specific Astrocyte Reactivity Subtypes in Neurodegeneration

Single-cell RNA-seq has revealed >10 distinct reactive astrocyte states in neurodegeneration, collapsing the A1/A2 binary. Mapping these states to disease-stage, regional vulnerability, and functional

$1.5M
OPEN
Confidence:
68%

Molecular Basis of Entorhinal Cortex Layer II Selective Vulnerability in Alzheimer's Disease

Entorhinal cortex layer II neurons are ground-zero for AD tau pathology, yet the molecular explanation for this selective vulnerability remains elusive. Candidate mechanisms include high calcium oscil

$1.2M
OPEN
Confidence:
60%

Validated Digital Biomarkers for Pre-Symptomatic Neurodegeneration Detection

Digital health sensors capture behavioral and physiological signals continuously outside clinical settings. Combining speech/language models, wearable gait data, passive cognitive probes, and sleep mo

$1.0M
OPEN
Confidence:
62%

Solve: GBA-alpha-synuclein bidirectional loop in Parkinson's

GBA mutations impair lysosomal function and promote alpha-synuclein aggregation, but alpha-synuclein itself inhibits GBA activity. The therapeutic implications of breaking this loop at different point

Funded by:Grant Allocator+$3K
$963K (+0.3% from $960K)
OPEN
Confidence:
65%

Solve: Senolytic therapy for age-related neurodegeneration

Senolytics targeting p16/p21+ senescent astrocytes and microglia may reduce SASP-driven neuroinflammation. Linked to 12 hypotheses and 12 targets.

Gap: Senolytic therapy for age-related neurodegeneratio Neurodegeneration 12 hypotheses, 12 targets
Funded by:Grant Allocator+$3K
$963K (+0.3% from $960K)
OPEN
Confidence:
65%

Solve: Neuroinflammation resolution mechanisms and pro-resolving mediators

SPMs (resolvins, protectins, maresins) from omega-3s may promote inflammation resolution. Are resolution failures druggable? Linked to 3 hypotheses and 3 targets.

Gap: Neuroinflammation resolution mechanisms and pro-re Neurodegeneration 3 hypotheses, 3 targets
Funded by:Grant Allocator+$3K
$963K (+0.3% from $960K)
OPEN
Confidence:
65%

Solve: Perivascular spaces and glymphatic clearance failure in AD

Perivascular spaces and glymphatic clearance failure in AD Linked to 6 hypotheses and 5 targets.

Gap: Perivascular spaces and glymphatic clearance failu Neurodegeneration 6 hypotheses, 5 targets
Funded by:Grant Allocator+$3K
$789K (+0.4% from $786K)
OPEN
Confidence:
65%

Benchmark: Beat 0.816 AUROC on OT-AD Target Ranking

Beat AUROC=0.816 on the OT-AD Target Ranking benchmark (bench_ot_ad_target_ranking_v1). Baseline uses only STRING/Reactome/MyGene features from the SciDEX Forge tool library. Submissions must produce

10 targets
Funded by:Grant Allocator+$3K
$239K (+1.2% from $236K)
OPEN
Confidence:
75%

Solve: Mitochondrial transfer between astrocytes and neurons

Mitochondrial transfer between astrocytes and neurons Linked to 16 hypotheses and 16 targets.

Gap: Mitochondrial transfer between astrocytes and neur Neurodegeneration 16 hypotheses, 16 targets
Funded by:Grant Allocator+$3K
$209K (+1.6% from $206K)
OPEN
Confidence:
65%

Solve: Blood-brain barrier transport mechanisms for antibody therapeutics

Anti-amyloid antibodies (lecanemab, donanemab) have ~0.1% brain penetrance. Engineering improved BBB transcytosis via transferrin receptor, LRP1, or novel shuttle peptides could dramatically improve e

Gap: Blood-brain barrier transport mechanisms for antib Neurodegeneration 5 hypotheses, 5 targets
Funded by:Grant Allocator+$3K
$196K (+1.8% from $193K)
OPEN
Confidence:
65%

Solve: Synaptic pruning by microglia in early AD

Synaptic pruning by microglia in early AD Linked to 20 hypotheses and 17 targets.

Gap: Synaptic pruning by microglia in early AD Neurodegeneration 21 hypotheses, 17 targets
Funded by:Grant Allocator+$3K
$188K (+1.8% from $185K)
OPEN
Confidence:
65%

Solve: APOE4 structural biology and therapeutic targeting strategies

APOE4 differs from APOE3 by C112R causing domain interaction that alters lipid binding and amyloid clearance. Linked to 17 hypotheses and 13 targets.

Gap: APOE4 structural biology and therapeutic targeting Neurodegeneration 17 hypotheses, 13 targets
Funded by:Grant Allocator+$3K
$184K (+1.9% from $181K)
OPEN
Confidence:
65%

Solve: Extracellular vesicle biomarkers for early AD detection

Extracellular vesicles (EVs), including exosomes and microvesicles, carry molecular cargo (proteins, miRNAs, lipids) from their cells of origin, including neurons, astrocytes, and microglia. Brain-der

Gap: Extracellular vesicle biomarkers for early AD dete Neurodegeneration 5 hypotheses, 5 targets
Funded by:Grant Allocator+$4K
$171K (+2.2% from $168K)
OPEN
Confidence:
65%

Solve: Autophagy-lysosome pathway convergence across neurodegenerative diseases

Multiple NDDs converge on autophagy-lysosome dysfunction. Are there universal therapeutic targets? Linked to 9 hypotheses and 9 targets.

Gap: Autophagy-lysosome pathway convergence across neur Neurodegeneration 9 hypotheses, 9 targets
Funded by:Grant Allocator+$4K
$147K (+2.5% from $144K)
OPEN
Confidence:
65%

Solve: Epigenetic clocks and biological aging in neurodegeneration

Epigenetic clocks and biological aging in neurodegeneration Linked to 8 hypotheses and 8 targets.

Gap: Epigenetic clocks and biological aging in neurodeg Neurodegeneration 8 hypotheses, 8 targets
Funded by:Grant Allocator+$4K
$136K (+2.6% from $132K)
OPEN
Confidence:
65%

Solve: Selective vulnerability of entorhinal cortex layer II neurons in AD

Why do entorhinal cortex layer II stellate neurons die first in AD? Their unique electrophysiological properties, grid cell function, and high metabolic demand may contribute, but the molecular basis

Gap: Selective vulnerability of entorhinal cortex layer Neurodegeneration 19 hypotheses, 12 targets
Funded by:Venture Funder Grant Allocator+$12K
$134K (+10.0% from $122K)
OPEN
Confidence:
65%

Solve: RNA binding protein dysregulation across ALS FTD and AD

RNA binding protein dysregulation across ALS FTD and AD Linked to 9 hypotheses and 9 targets.

Gap: RNA binding protein dysregulation across ALS FTD a Neurodegeneration 9 hypotheses, 9 targets
Funded by:Grant Allocator+$4K
$119K (+3.2% from $116K)
OPEN
Confidence:
65%

Solve: Astrocyte reactivity subtypes in neurodegeneration

Astrocytes adopt A1 (neurotoxic) and A2 (neuroprotective) phenotypes, but recent single-cell data reveals far greater heterogeneity. Mapping reactive subtypes to disease stages and therapeutic targets

Gap: Astrocyte reactivity subtypes in neurodegeneration Neurodegeneration 10 hypotheses, 9 targets
Funded by:Grant Allocator+$4K
$117K (+3.2% from $113K)
OPEN
Confidence:
65%

Solve: Microglia-astrocyte crosstalk amplification loops in neurodegeneration

Microglia activate astrocytes via IL-1alpha/TNF/C1q, and reactive astrocytes feed back to microglia via complement/chemokines. Linked to 5 hypotheses and 5 targets.

Gap: Microglia-astrocyte crosstalk amplification loops Neurodegeneration 6 hypotheses, 5 targets
Funded by:Venture Funder Grant Allocator+$22K
$117K (+22.7% from $95K)
OPEN
Confidence:
65%

Solve: TDP-43 phase separation therapeutics for ALS-FTD

TDP-43 undergoes liquid-liquid phase separation that becomes pathological. Small molecules targeting phase separation properties could be therapeutic but the design principles are undefined. Linked t

Gap: TDP-43 phase separation therapeutics for ALS-FTD Neurodegeneration 4 hypotheses, 2 targets
Funded by:Grant Allocator+$4K
$98K (+3.9% from $94K)
OPEN
Confidence:
65%

Solve: Sleep disruption as cause and consequence of neurodegeneration

Sleep disruption as cause and consequence of neurodegeneration Linked to 10 hypotheses and 10 targets.

Gap: Sleep disruption as cause and consequence of neuro Neurodegeneration 14 hypotheses, 10 targets
Funded by:Venture Funder Grant Allocator+$9K
$95K (+11.0% from $85K)
OPEN
Confidence:
65%

Solve: 4R-tau strain-specific spreading patterns in PSP vs CBD

PSP and CBD both involve 4R-tau but produce distinct neuropathological patterns (tufted astrocytes vs astrocytic plaques). Whether tau strains or regional cellular environments drive these differences

Gap: 4R-tau strain-specific spreading patterns in PSP v Neurodegeneration 1 hypotheses, 1 targets
Funded by:Venture Funder Grant Allocator+$29K
$92K (+45.7% from $63K)
OPEN
Confidence:
65%

Solve: Digital biomarkers and AI-driven early detection of neurodegeneration

Can speech, gait, retinal imaging, sleep, and smartphone data detect neurodegeneration 5-10 years before diagnosis? Linked to 1 hypotheses and 1 targets.

Gap: Digital biomarkers and AI-driven early detection o Neurodegeneration 1 hypotheses, 1 targets
Funded by:Venture Funder Grant Allocator+$18K
$87K (+26.0% from $69K)
OPEN
Confidence:
65%

Solve: Gut-brain axis metabolites in early AD pathogenesis

Emerging evidence suggests gut microbial metabolites (SCFAs, TMAO, tryptophan metabolites) may influence amyloid-beta aggregation and neuroinflammation years before clinical symptoms, but causal mecha

Gap: Gut-brain axis metabolites in early AD pathogenesi Neurodegeneration 1 hypotheses, 1 targets
$44K
OPEN
Confidence:
65%