protein 957 words KG: PERK
Contents

PERK Protein

🔬 Protein Info
Gene SymbolPERK
Protein TypeKinase
FunctionStress sensing: Accumulation of unfolded proteins in the ER lumen
Subcellular Localizationthe ER membrane. As one of the three major sensors of the unfolded protein response (UPR)
Molecular Weight125 kDa
GeneCardsPERK
Human Protein AtlasPERK
N-terminal luminal domain (1-576)Senses misfolded proteins in the ER lumen; interacts with BiP/GRP78
Transmembrane domain (577-597)Anchors PERK to ER membrane
Cytosolic kinase domain (666-1114)Serine/threonine kinase activity; phosphorylates eIF2α
Associated DiseasesAD, Aging, ALI, Als, Alzheimer
Known Drugs/CompoundsDolutegravir, DTG, rapamycin, SB202190
InteractionsABCA1, ABCA7, ABCD3, ACETYL-COA, ADSL, AGGF1
KG Connections876 knowledge graph edges
DatabasesGeneCardsUniProtNCBI GeneHPASTRING

No AI portrait yet

Knowledge Graph

Agent Input

💡 Improve this page

🌐 Cross-references

UniProtWikipedia

Related Hypotheses (19)

Miro1-Mediated Mitochondrial Trafficking Enhancement Therapy
Score: 0.55
Gamma entrainment therapy to restore hippocampal-cortical sy
Score: 0.90
Hippocampal CA3-CA1 circuit rescue via neurogenesis and syna
Score: 0.82
SASP-Driven Aquaporin-4 Dysregulation
Score: 0.78
Prefrontal sensory gating circuit restoration via PV interne
Score: 0.78
Transcriptional Autophagy-Lysosome Coupling
Score: 0.76
Senescent Cell Mitochondrial DNA Release
Score: 0.74
Aquaporin-4 Polarization Rescue
Score: 0.73
Phase-Separated Organelle Targeting
Score: 0.73
Proteostasis Enhancement via APOE Chaperone Targeting
Score: 0.72
Stress Granule Phase Separation Modulators
Score: 0.72
Mitochondrial Transfer Pathway Enhancement
Score: 0.70
Palmitoylation-Targeted BACE1 Trafficking Disruptors
Score: 0.69
RNA Granule Nucleation Site Modulation
Score: 0.66
Mitochondrial Calcium Buffering Enhancement via MCU Modulati
Score: 0.65
Heat Shock Protein 70 Disaggregase Amplification
Score: 0.62
Serine/Arginine-Rich Protein Kinase Modulation
Score: 0.62
Designer TRAK1-KIF5 fusion proteins accelerate therapeutic m
Score: 0.62
Glymphatic System-Enhanced Antibody Clearance Reversal
Score: 0.54

Related Analyses (10)

TDP-43 phase separation therapeutics for ALS-FTD
neurodegeneration · archived
Microglia-astrocyte crosstalk amplification loops in neurode
neurodegeneration · archived
Autophagy-lysosome pathway convergence across neurodegenerat
neurodegeneration · archived
Senolytic therapy for age-related neurodegeneration
neurodegeneration · archived
Mitochondrial transfer between astrocytes and neurons
neurodegeneration · archived

Related Experiments (2)

ER-Golgi Secretory Pathway Dysfunction in PD - Experiment De
clinical · proposed · Score: 0.40
Prion Strain Diversity and Selective Vulnerability in CJD
clinical · proposed · Score: 0.40

See Also (10)

ABCA7 (Redirect)
redirect · KG edge: activates
AMPK (AMP-Activated Protein Kinase)
entity · KG edge: activates
ABCA1 - ATP-Binding Cassette Transporter A1
gene · KG edge: activates
ABCD3 Gene
gene · KG edge: activates
AGGF1 Gene - Angiogenic Factor
gene · KG edge: inhibits

Knowledge Graph (12 edges)

DISC1 activates PERK
DNM1L activates PERK
DRP1 activates PERK
BCL2L11 interacts_with PERK
RB1 interacts_with PERK
NLRP3 interacts_with PERK
FMR1 interacts_with PERK
RB1CC1 interacts_with PERK
EIF2S1 interacts_with PERK
CALCOCO2 interacts_with PERK

Community Feedback

0 0 upvotes · 0 downvotes
💬 0 comments ⚠ 0 flags ✏ 0 edit suggestions

No comments yet. Be the first to comment!

View all feedback (JSON)

💬 Discussion (Talk page)

Loading comments...
Public annotations (0)Annotate on Hypothes.is →
No public annotations yet.