gene 1,814 words KG: CGAS
Contents

CGAS Gene

🧬 Gene Info
Gene SymbolCGAS
Chromosome6q15
Protein TypeEnzyme
Target ClassEnzyme
FunctionSmall molecule inhibitor of cyclic dinucleotide synthesis
Mechanism of ActionSmall molecule inhibitor of cyclic dinucleotide synthesis
DruggabilityMedium (0.47)
Clinical StagePhase III
Molecular Weight57 kDa
Amino Acids522 aa
Exons8
PathwaysAkt, Amyloid, Apoptosis, Autophagy, Calcium Signaling
UniProt IDQ8N884
NCBI Gene ID115004
Ensembl IDENSG00000154122
GeneCardsCGAS
Human Protein AtlasCGAS
Associated Diseasesaging, Als, Alzheimer
Known Drugs/CompoundsAberrant DNA, cGAS Inhibitors, Ginkgetin, Mitochondrial Dna, Mitochondrial DNA, mtDNA
InteractionsACHE, Actin, AD, AGING, AHR, AKT
SciDEX TargetView Target Profile (4 clinical trials)
KG Connections1976 knowledge graph edges
DatabasesGeneCardsHPASTRING

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🌐 Cross-references

NCBI GeneUniProtGeneCardsWikipediaHGNCEnsembl

Related Hypotheses (50)

Senescent Cell Mitochondrial DNA Release
Score: 0.74
Selective APOE4 Degradation via Proteolysis Targeting Chimer
Score: 0.79
Competitive APOE4 Domain Stabilization Peptides
Score: 0.78
Selective HDAC3 Inhibition with Cognitive Enhancement
Score: 0.78
Chromatin Accessibility Restoration via BRD4 Modulation
Score: 0.77
APOE4 Allosteric Rescue via Small Molecule Chaperones
Score: 0.76
Cell-Type Specific TREM2 Upregulation in DAM Microglia
Score: 0.76
Targeted APOE4-to-APOE3 Base Editing Therapy
Score: 0.76
GFAP-Positive Reactive Astrocyte Subtype Delineation
Score: 0.75
APOE Isoform Expression Across Glial Subtypes
Score: 0.74
Epigenetic Memory Erasure via TET2 Activation
Score: 0.74
PARP1 Inhibition Therapy
Score: 0.74
SIRT3-Mediated Mitochondrial Deacetylation Failure with PINK
Score: 0.74
Aquaporin-4 Polarization Rescue
Score: 0.73
CYP46A1 Overexpression Gene Therapy
Score: 0.73
Phase-Separated Organelle Targeting
Score: 0.73
TFAM overexpression creates mitochondrial donor-recipient gr
Score: 0.73
Interfacial Lipid Mimetics to Disrupt Domain Interaction
Score: 0.72
Circadian Rhythm Entrainment of Reactive Astrocytes
Score: 0.72
Astroglial Gap Junction Coordination via Connexin-43 Phospho
Score: 0.72
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Related Analyses (21)

Gene expression changes in aging mouse brain predicting neur
neurodegeneration · completed
Senolytic therapy for age-related neurodegeneration
neurodegeneration · archived
Microglia-astrocyte crosstalk amplification loops in neurode
neurodegeneration · archived
Autophagy-lysosome pathway convergence across neurodegenerat
neurodegeneration · archived
Neuroinflammation resolution mechanisms and pro-resolving me
neurodegeneration · archived

Related Experiments (4)

cGAS/STING pathway activation by TDP-43-released mtDNA
exploratory · proposed · Score: 0.95
Sporadic ALS Initiation Biology: Deep Phenotyping of At-Risk
clinical · proposed · Score: 0.40
cGAS-STING Pathway Validation Study in Parkinson's Disease
clinical · proposed · Score: 0.40
Proposed experiment from debate on Senolytics targeting p16/
falsification · proposed · Score: 0.40

See Also (3)

AKT1 Gene
gene · KG edge: regulates
Packard Center for ALS Research
institution · KG edge: activates
Aging vs Neurodegeneration: Mechanistic Comparison Matr
mechanism · KG edge: activates

Knowledge Graph (12 edges)

CGAS associated_with neurodegeneration
CGAS interacts_with STING1
CGAS interacts_with DNASE2
STING1 interacts_with CGAS
DNASE2 interacts_with CGAS
MMP9 co_discussed CGAS
SLC7A11 co_discussed CGAS
CGAS co_discussed AQP4
CGAS co_discussed CD38
CGAS co_discussed C1Q

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