entity

PARP

Entity Detail — Knowledge Graph Node

Understanding Entity Pages

This page aggregates everything SciDEX knows about PARP: its mechanistic relationships (Knowledge Graph edges), hypotheses targeting it, analyses mentioning it, and supporting scientific papers. The interactive graph below shows its immediate neighbors. All content is AI-synthesized from peer-reviewed literature.

8Connections
3Hypotheses
1Analyses
6Outgoing
2Incoming
2Experiments
1Debates

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Wiki Pages (13)

Knowledge base pages for this entity

Canonical Page

PARP Inhibitor Therapy for Neurodegeneration

idea · 956 words

PARP Inhibitor Therapy

therapeutic · 1769 words

PARP in Neurodegeneration

mechanism · 1341 words

Synthetic Lethality and PARP Inhibition in Neurodegeneration

mechanism · 1295 words

PARP4 — Poly(ADP-Ribose) Polymerase 4

gene · 1115 words

PARP1 Inhibition for Parthanatos Prevention in Neurodegeneration

idea · 1069 words

Outgoing (6)

TargetRelationTypeStr
DNA Damage/Repairinvolved_inprocess0.90
ADP Ribosylationcatalyzesprocess0.90
DNA Repairinvolved_inprocess0.90
DNA Damage/Repaircatalyzesprocess0.88
NAD+degradeschemical0.80

Incoming (2)

SourceRelationTypeStr
Nad+regulatescompound0.95
Parp Inhibitorstrapsdrug0.90

Targeting Hypotheses (3)

Hypotheses where this entity is a therapeutic target

HypothesisScoreDiseaseAnalysis
PARP1-NAD+-AIF bioenergetic collapse drives a self-amplifyin 0.760 neurodegeneration What mechanisms drive the self-amplifyin
PARP1 Inhibition Therapy 0.738 neurodegeneration TDP-43 phase separation therapeutics for
PARP1 Inhibition Blocks Poly(PR)-Triggered DNA Damage and Su 0.661 neurodegeneration What upstream mechanisms trigger p53 act

Mentioning Analyses (1)

Scientific analyses that reference this entity

Do oligodendrocytes require DNA repair enhancement or inhibition for neuroprotec

neurodegeneration | 2026-04-11 | 0 hypotheses

Experiments (2)

Experimental studies targeting or related to this entity

ExperimentTypeDiseaseScoreFeasibilityModelStatusEst. Cost
DNA Damage Repair Deficiency Validation Study in Parkinson's Disease clinical Parkinson's Disease 0.400 0.50 human completed $7,500,000
Regulated Necrosis Validation Study in Parkinson's Disease clinical Parkinson's Disease 0.400 0.50 human proposed $6,550,000

Related Papers (20)

Scientific publications cited in analyses involving this entity

Title & PMIDAuthorsJournalYearCitations
Transcription-replication conflicts underlie sensitivity to PARP inhibitors. [PMID:38509368] Petropoulos M, Karamichali A, Rossetti G Nature 2024 1
PARP1-DOT1L transcription axis drives acquired resistance to PARP inhibitor in o [PMID:38778348] Liu C, Li J, Xu F, Chen L, Ni M, Wu J, Z Mol Cancer 2024 1
USP1 deubiquitinates PARP1 to regulate its trapping and PARylation activity. [PMID:39536107] Nespolo A, Stefenatti L, Pellarin I, Gam Sci Adv 2024 1
NAD(+) rescues aging-induced blood-brain barrier damage via the CX43-PARP1 axis. [PMID:37683629] Zhan R, Meng X, Tian D, Xu J, Cui H, Yan Neuron 2023 1
Nuclear cGAS suppresses DNA repair and promotes tumorigenesis. [PMID:30356214] Liu H, Zhang H, Wu X, Ma D, Wu J, Wang L Nature 2018 1
Defective DNA Damage Response Is a Targetable Therapeutic Vulnerability in ESR1- [PMID:41499130] Herzog SK, Stevens JH, Gu G, Grimm SL, C Cancer Res 2026 0
Replicative gaps in DNA damage tolerance, genome instability, and cancer therapy [PMID:41864203] Falbo L, Costanzo V Mol Cell 2026 0
Versatile and sensitive detection of mono- and poly(ADP-ribosyl)ation reveals XR [PMID:41922367] Dauben H, Mihaljević M, Kolvenbach A, Pa Nat Commun 2026 0
Differential proteomic responses to short-term heat stress in Vechur and crossbr [PMID:41931203] Anisha J P; Shynu M; Radhika G; Beena V; Tropical animal health and pro 2026 0
Differential sensitivity of MCPH1- and BRCA2-deficient cancer cells to PARP-1 in [PMID:41931484] Chapman IG, Wu X, Veuger S, Jowsey PA PLoS One 2026 0
Targeting Poly (ADP-Ribose) Polymerase-1 for the Treatment of Neurodegenerative [PMID:41178110] Polk S, Rassaeikashuk M, Thilagavathi R, Chemical biology & drug design 2025 0
Increased nucleotide metabolism alleviates Alzheimer's disease pathology. [PMID:41102145] ["Yu Y", "Miller M", "Huang A", "Tan B", Cell death & disease 2025 0
Roles and therapeutic potential of PARP-1 in neurodegenerative diseases. [PMID:41022359] ["Liu C", "Lai F", "Zhang T", "Mao K", " Biochemical pharmacology 2025 0
Tipping the PARylation scale: Dysregulation of PAR signaling in Huntington and n [PMID:40905723] Peng C, Maiuri T, Truant R Journal of Huntington's diseas 2025 0
Targeting KCNN4 channels modulates microglial activation and apoptosis in a PD-r [PMID:40913912] ["Hung H", "Li I", "Lin Y", "Yeh T", "Ng Biomedicine & pharmacotherapy 2025 0
Clinical approaches to overcome PARP inhibitor resistance. [PMID:40442774] ["Zou Y", "Zhang H", "Chen P", "Tang J", Molecular cancer 2025 0
PARPs and PARP inhibitors: molecular mechanisms and clinical applications. [PMID:41460301] Wang F, Guo Z, Carr MJ, Shi W Molecular biomedicine 2025 0
Efficacy of Adding Veliparib to Temozolomide for Patients With MGMT-Methylated G [PMID:39480453] ["Sarkaria J", "Ballman K", "Kizilbash S JAMA oncology 2024 0
PARP Inhibitors for Breast Cancer Treatment: A Review. [PMID:38512229] ["Morganti S", "Marra A", "De Angelis C" JAMA oncology 2024 0
Blocking the Self-Destruct Program of Dopamine Neurons through Macrophage Migrat [PMID:38396375] ["Patel J", "Dawson V", "Dawson T"] Movement disorders : official 2024 0

Debates (1)

Multi-agent debates referencing this entity

The debate revealed conflicting therapeutic approaches - enhancing DNA repair ve

closed · Rounds: 4 · Score: 1.00 · 2026-04-20

Related Research

Hypotheses and analyses mentioning PARP in their description or question text

No additional research found