Silibinin-induced G2/M cell cycle arrest in breast cancer cells

Exploratory Score: 0.900 Price: $0.50 breast cancer MCF-7 and MDA-MB-231 human breast cancer cell lines Status: proposed

What This Experiment Tests

Exploratory experiment designed to discover new patterns targeting YAP1, CAPZA1 in MCF-7 and MDA-MB-231 human breast cancer cell lines. Primary outcome: G2/M cell cycle arrest and F-actin disassembly

Description

This experiment investigated the mechanism by which silibinin induces cell cycle arrest in breast cancer cells. The study examined both hormone-sensitive MCF-7 and triple-negative MDA-MB-231 breast cancer cells to determine how silibinin treatment affects cell cycle progression. The researchers found that silibinin induces G2/M phase arrest in both cell lines through inhibition of the YAP pathway. Additionally, they discovered that silibinin significantly reduces F-actin assembly, which is positively regulated by YAP through transcriptional control of polymerization factors. The study demonstrated that F-actin disassembly is not merely a consequence of YAP inhibition but actively contributes to cell cycle arrest. Using molecular techniques including siRNA transfection and cytoskeletal disruption with Cytochalasin D, they showed that F-actin assembly disturbance directly contributes to cell cycle arrest independent of YAP activity.

TARGET GENE
YAP1, CAPZA1
MODEL SYSTEM
MCF-7 and MDA-MB-231 human breast cancer cell lines
ESTIMATED COST
$0
TIMELINE
0 months
PATHWAY
YAP signaling, actin cytoskeleton organization, cell cycle regulation
SOURCE
extracted_from_pmid_41349910
PRIMARY OUTCOME
G2/M cell cycle arrest and F-actin disassembly

Scoring Dimensions

Info Gain 0.00 (25%) Feasibility 0.00 (20%) Hyp Coverage 0.00 (20%) Cost Effect. 0.00 (15%) Novelty 0.00 (10%) Ethical Safety 0.00 (10%) 0.900 composite

📖 Wiki Pages

YAP1 — Yes-Associated Protein 1geneYAP1 ProteinproteinYAP/TAZ (Hippo) Signaling in NeurodegenerationmechanismYAP/TAZ Signaling Pathway in NeurodegenerationmechanismYAP/TAZ Mechanoactivation Protocol for NeurodegeneideaYAP/TEAD Pathway Modulators for NeurodegenerationtherapeuticCancerdiseaseCancerdiseaseResearchersindexHippo Signaling in 4R-TauopathiesmechanismHippo Signaling Pathway in Parkinson's Diseasemechanism

Protocol

Cell culture, silibinin treatment, cell cycle analysis, F-actin staining and microscopy, siRNA transfection (si-YAP/TAZ, si-Capza1), Cytochalasin D treatment, qRT-PCR, protein analysis

Expected Outcomes

Silibinin treatment expected to induce cell cycle arrest through YAP inhibition; discovered that F-actin disassembly is a critical mediator of this effect

Success Criteria

Demonstration of G2/M arrest, reduced F-actin assembly, and restoration of cell cycle progression upon F-actin stabilization

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