FK866 in azoxymethane/DSS colitis-associated cancer model

Validation Score: 0.850 Price: $0.50 Colitis-associated cancer AOM/DSS-treated mice Status: proposed

What This Experiment Tests

Validation experiment designed to validate causal mechanisms targeting NAMPT in AOM/DSS-treated mice. Primary outcome: Tumor development and inflammatory markers

Description

Evaluation of FK866's therapeutic potential in preventing inflammation-associated tumorigenesis using the azoxymethane (AOM)/DSS model of colitis-associated cancer in mice. This experiment assessed whether NAMPT inhibition could suppress both inflammatory processes and tumor development in the context of chronic intestinal inflammation. The study demonstrated that FK866 treatment effectively suppressed inflammation-associated tumorigenesis, indicating that NAD metabolism plays a crucial role not only in acute inflammation but also in the progression from chronic inflammation to cancer.

TARGET GENE
MODEL SYSTEM
AOM/DSS-treated mice
ESTIMATED COST
$0
TIMELINE
0 months
PATHWAY
NAD salvage pathway, inflammation-cancer axis
SOURCE
extracted_from_pmid_28877980
PRIMARY OUTCOME
Tumor development and inflammatory markers

Scoring Dimensions

Info Gain 0.00 (25%) Feasibility 0.00 (20%) Hyp Coverage 0.00 (20%) Cost Effect. 0.00 (15%) Novelty 0.00 (10%) Ethical Safety 0.00 (10%) 0.850 composite

📖 Wiki Pages

NAMPT ProteinproteinNAMPT GenegeneNAD+ Boosters for NeurodegenerationtherapeuticNAD+ Precursors for Neurodegenerationtherapeuticnad-augmentation-therapy-early-adgeneralNAD+ Precursors (NMN/NR) for Parkinson's DiseasetherapeuticNAD+ Precursor Therapy for Neurodegenerative DiseatherapeuticNAD+ Bioenergetics Investment SynthesismechanismNAD+ Metabolism in NeurodegenerationmechanismNAD+ Metabolism Pathway in NeurodegenerationmechanismNAD Signaling in NeurodegenerationmechanismNAD Kinase ProteinproteinNAD+ Boosters for NeurodegenerationtherapeuticCancerdiseaseCancerdisease

Protocol

Sequential AOM and DSS treatment to induce colitis-associated cancer followed by FK866 intervention with assessment of tumor formation and inflammatory parameters

Expected Outcomes

Reduced tumor formation and suppressed inflammatory tumorigenesis

Success Criteria

Decreased tumor incidence and size, reduced inflammatory markers

Related Hypotheses (3)

TREM2 R47H Variant-Driven Metabolic Dysfunction as the Primary Trigger for Failed DAM Transition0.862
Metabolic NAD+ Salvage Pathway Enhancement Through NAMPT Overexpression0.745
NAD+ Salvage Pathway Optimization0.455

Debate History (0)

No debates yet

Experiment Results (0)

No results recorded yet. Use POST /api/experiments/{id}/results to record a result.